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TBD from US Patent US20240059694: "COMPOUND CONTAINING 1,3-BENZODIOXOL STRUCTURE AND PREPARATION METHOD AND USE THEREOF"
Assay data:28 Active, 30 Activity ≤ 1 µM, 30 Tested
SummaryRelated BioAssays by Target
Determination of Related Protease Inhibition from US Patent US20240059691: "ENZYME INHIBITORS"
Assay data:279 Active, 16 Activity ≤ 1 nM, 253 Activity ≤ 1 µM, 299 Tested
THR/RXR Heterodimer Assay for Thyroid Hormone Receptor Agonist Screening from US Patent US20240059682: "THYROID HORMONE RECEPTOR BETA AGONIST COMPOUNDS"
Assay data:26 Active, 25 Activity ≤ 1 µM, 26 Tested
Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) Assay for Thyroid Hormone Receptor Agonist Screening from US Patent US20240059682: "THYROID HORMONE RECEPTOR BETA AGONIST COMPOUNDS"
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
THR Reporter Gene Method from US Patent US20240059676: "THYROID HORMONE RECEPTOR b SELECTIVE AGONIST COMPOUND, PHARMACEUTICAL COMPOSITION AND USE THEREOF"
Assay data:32 Active, 21 Activity ≤ 1 µM, 38 Tested
Biochemical QPCT and QPCTL Activity Assay from US Patent US20240059675: "PIPERIDINYLPYRIDINYLCARBONITRILE DERIVATIVES AS INHIBITORS OF GLUTAMINYL-PEPTIDE CYCLOTRANSFERASE AND GLUTAMINYL-PEPTIDE CYCLOTRANSFERASE LIKE PROTEIN"
Assay data:36 Active, 8 Activity ≤ 1 nM, 36 Activity ≤ 1 µM, 36 Tested
In Vitro Kinase Binding Assay from US Patent US20240058459: "DENDRIMER COMPOSITIONS AND METHODS FOR DRUG DELIVERY TO THE EYE"
Assay data:3 Active, 2 Activity ≤ 1 nM, 3 Activity ≤ 1 µM, 3 Tested
In Vitro JAK Kinase Assay from US Patent US20240058343: "TREATMENT OF URTICARIA USING JAK INHIBITORS"
Assay data:26 Active, 26 Activity ≤ 1 µM, 26 Tested
Measuring Antiviral Effect of Compounds from US Patent US11905306: "Substituted phenyl ethynyl pyridine carboxamides as potent inhibitors of SARS virus"
Assay data:70 Active, 38 Activity ≤ 1 µM, 80 Tested
Biochemical EC50 Assay from US Patent US20240050576: "METHODS AND COMPOUNDS FOR THE TREATMENT OF GENETIC DISEASE"
Assay data:51 Active, 61 Activity ≤ 1 µM, 61 Tested
Assay for Inhibition of MMP from US Patent US20240050571: "CARBORANE HYDROXAMIC ACID MATRIX METALLOPROTEINASE INHIBITORS AND AGENTS FOR BORON NEUTRON CAPTURE THERAPY"
Assay data:4 Active, 1 Activity ≤ 1 nM, 4 Activity ≤ 1 µM, 4 Tested
IC50 Determination from US Patent US20240043470: "MACROCYCLIC COMPOUNDS AS PROTEASOME INHIBITORS"
Assay data:80 Active, 18 Activity ≤ 1 µM, 160 Tested
MCF-7 Cell Growth Study from US Patent US20240043442: "SELECTIVE ESTROGEN RECEPTOR DEGRADERS AND USES THEREOF"
Assay data:50 Active, 30 Activity ≤ 1 nM, 50 Activity ≤ 1 µM, 50 Tested
Antiviral Assay from US Patent US20240043417: "COMPOUNDS FOR THE TREATMENT OF SARS"
Assay data:1 Active, 19 Tested
SARS-CoV-2 3CLpro Enzyme Assay from US Patent US20240043417: "COMPOUNDS FOR THE TREATMENT OF SARS"
Assay data:11 Active, 23 Tested
Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) Assay from US Patent US20240043404: "APOPTOSIS INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES"
Assay data:372 Active, 356 Activity ≤ 1 nM, 372 Activity ≤ 1 µM, 372 Tested
Determination of the Effect of a SERCA Agonist on the Reduction of ER Stress from US Patent US11890279: "Quinolines that modulate SERCA and their use for treating disease"
Assay data:11 Tested
TBD from US Patent US20240034743: "TRICYCLIC COMPOUNDS AS EGFR INHIBITORS"
Assay data:135 Active, 118 Activity ≤ 1 nM, 137 Activity ≤ 1 µM, 137 Tested
Assay data:133 Active, 31 Activity ≤ 1 nM, 137 Activity ≤ 1 µM, 137 Tested
CDK2/Cyclin E1 Full length ADP-Glo Kinase Assay from US Patent US20240034731: "AZA-QUINAZOLINE COMPOUNDS AND METHODS OF USE"
Assay data:95 Active, 92 Activity ≤ 1 µM, 97 Tested
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