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Chemical stability of the compound assessed as acid-catalyzed hydrolysis by measuring rate constant
Assay data:7 Tested
Summary
Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK cell membrane at 10 uM incubated for 30 mins by microplate beta scintillation counting based radioligand inhibition assay relative to control
Assay data:5 Tested
SummaryPubMed CitationRelated BioAssays by Target
Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane at 10 uM incubated for 60 mins by microplate beta scintillation counting based radioligand inhibition assay relative to control
Assay data:9 Tested
Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cell membrane ay 10 uM incubated for 30 mins by microplate beta scintillation counting based radioligand inhibition assay relative to control
Assay data:13 Tested
Displacement of [3H]NECA from human adenosine A3 receptor expressed in HeLa cell membrane at 10 uM incubated for 180 mins by microplate beta scintillation counting based radioligand inhibition assay relative to control
Assay data:6 Tested
ERK5 transcriptional activity HTS
Assay data:60 Active, 2000 Tested
SummaryCompounds, ActivePubMed Citation
qHTS Assay for Inhibitors of N-terminal methyltransferase 1 (NTMT1): MTaseGlo Assay Confirmatory Screen, Round 1
Assay data:7 Active, 258 Tested
SummaryCompounds, ActiveRelated BioAssays by Depositor
qHTS Assay for Inhibitors of N-terminal methyltransferase 1 (NTMT1): ThioGlo Assay Confirmatory Screen, Round 2
Assay data:125 Active, 258 Tested
SummaryCompounds, ActiveRelated BioAssays by DepositorRelated BioAssays by Target
qHTS Assay for Inhibitors of N-terminal methyltransferase 1 (NTMT1): ThioGlo3 Assay Confirmatory Screen, Round 1.
qHTS assay for MDR1-selective chemotherapeutics: Primary screen using the drug-selected MDR subline cells KB-V1
Assay data:13449 Active, 399619 Tested
qHTS assay for MDR1-selective chemotherapeutics: Primary screen using the parental adenocarcinoma cell KB-3-1
Assay data:5540 Active, 399561 Tested
qHTS assay for inhibitors of human lactate dehydrogenase
Assay data:736 Active, 484712 Tested
SSB-PriA antibiotic resistant target AlphaScreen
Assay data:2577 Active, 432182 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
GENE-TOX mutagenicity studies
Assay data:1995 Active, 3214 Tested
SummaryCompounds, Active
CCRIS mutagenicity studies
Assay data:4929 Active, 8266 Tested
Cytotoxicity against human MCF7 cells assessed as inhibition of cell viability after 48 hrs by MTT assay
Assay data:8 Tested
Cytotoxicity against rat C6 cells assessed as inhibition of cell viability after 48 hrs by MTT assay
Cytotoxicity against human DU145 cells assessed as inhibition of cell viability after 48 hrs by MTT assay
Cytotoxicity against human HaCaT cells assessed as inhibition of cell viability after 48 hrs by MTT assay
Cytotoxicity against rat L6 cells assessed as inhibition of cell viability after 48 hrs by MTT assay
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